参考文献/References:
[1]MAES B U W. Topics in heterocyclic chemistry: Vol.26 [M]. Berlin: Springer-Verlag, 2010.
[2]SHIRI M. Indoles in multicomponent processes(MCPs)[J]. Chem Rev, 2012, 112(6): 3508-3549.
[3]ROMAGNOLI R, BARALDI P G, SARKAR T,et al. Synthesis and Biological Evaluation of 1-Methyl-2-(3',4',5'-trimethoxybenzoyl)-3-aminoindoles as a New Class of Antimitotic Agents and Tubulin Inhibitors[J]. J Med Chem, 2008, 51(5): 1464-1468.
[4]BRANCALEA, SILVESTRI R. Indole, a core nucleus for potent inhibitors of tubulin polymerization[J]. Med Res Rev, 2007, 27(2): 209-238.
[5]MAHBOOBIS, SELLMER A, HOÖCHER H, et al. 2-Aroylindoles and 2-Aroylbenzofurans with N-Hydroxyacrylamide Substructures as a Novel Series of Rationally Designed Histone Deacetylase Inhibitors[J]. J Med Chem, 2007, 50(18): 4405-4418.
[6]WILLSONT M, BROWN P J, STERNBACH D D, et al. The PPARs: from orphan receptors to drug discovery[J]. J Med Chem, 2000, 43(4): 527-550.
[7]CRUZ-LÓPEZ O, DÍAZ-MOCHÓ J J, CAMPOS J M, et al. Design, syntheses, biological evaluation, and docking studies of 2-substituted 5-methylsulfonyl-1-phenyl-1H-indoles: potent and selective in vitro cyclooxygenase-2 inhibitors[J]. ChemMedChem, 2007, 2(1): 88-100.
[8]MAHBOOBI S, TELLER S, PONGRATZ H,et al. Bis(1H-2-indolyl)methanones as a novel class of inhibitors of the platelet-derived growth factor receptor kinase[J]. J Med Chem, 2002, 45(5): 1002-1008.
[9]OKAUCHI T, ITONAGA M, MINAMI T, et al. A general method for acylation of indoles at the 3-position with acyl chlorides in the presence of dialkylaluminum chloride[J]. Org Lett, 2000, 2(10): 1485-1487.
[10]GUCHHAIT S K, KASHYAP M, KAMBLE H. ZrCl4-mediated regio- and chemoselective friedel-crafts acylation of indole[J]. J Org Chem, 2011, 76(11): 4753-4758.
[11]KATRITSKY A R, AKUTAGAWA K.Carbon dioxide: a reagent for the protection of nucleophilic centres and the simultaneous activation of alternative locations to electrophilic attack: Part I, new synthetic method for the 2-substitution of 1-unsubstituted indoles[J]. Tetrahedron Lett, 1985, 26(48): 5935-5938.
[12]GHARPURE M, STOLLER A, BELLAMY F. The N-tert-butylcarbamoyl directed metalation group for the regiospecific synthesis of 2-substituted pyrroles and indoles[J]. Synthesis, 1991(12): 1079-1082.
[13]YANG Q Q, XIAO C, LU L Q. et al. Synthesis of indoles through highly efficient cascade reactions of sulfur ylides and N-(ortho-chloromethyl)aryl amides[J]. Angew Chem Int Ed, 2012, 51(36): 9137-9140.
[14]GORIYA Y, RAMANA C V.2-Aroylindoles from o-bromochalcones via Cu(I)-catalyzed SNAr with an azide and intramolecular nitrene C-H insertion[J]. Chem Commun, 2014, 50(58): 7790-7792.
[15]OKURO K, GURNHAM J, ALPER H. Ionic diamine rhodium complex catalyzed reductive N-heterocyclization of 2-nitrovinylarenes[J]. J Org Chem, 2011, 76(11): 4715-4720.
[16]YANG K, ZHOU F, KUANG Z, et al. Diborane-mediated deoxygenation of o-nitrostyrenes to form indoles[J]. Org Lett, 2016, 18(16): 4088-4091.
[17]ZHAO Y, LI D, ZHAO L, et al. A practical synthesis of 2-aroylindoles from N-(2-formylphenyl)trifluoro-acetamides in PEG-400[J]. Synthesis, 2011, 6: 873-880.
[18]ZHOU B, YANG Y, LI Y. Rhodium-catalyzed oxidative C2-acylation of indoles with aryl and alkyl aldehydes[J]. Chem Commun, 2012, 48(42): 5163-5165.
[19]KUMAR G, SEKAR G. Pd-catalyzed direct C2-acylation and C2, C7-diacylation of indoles: pyrimidine as an easily removable C—H directing group[J]. RSC Adv, 2015, 5(36): 28292-28298.
[20]CAI S, LIN S, YI X. Substrate-controlled transformation of azobenzenes to indazoles and indoles via Rh(III)-catalysis[J]. J Org Chem, 2017, 82(1): 512-520.
[21]BLACK D S C, WONG L C H.A simple synthesis of 2-acyl indoles from isatins[J]. J Chem Soc Chem Commun, 1980(4): 200-200.
[22]RAMKUMAR N, NAGARAJAN R. A new route to the synthesis of ellipticine quinone from isatin[J]. Tetrahedron Lett, 2014, 55(5): 1104-1106.
[23]SHMIDT M S, PERILLO I A, CAMELLI A,et al. Polyfunctional 4-quinolinones. Synthesis of 2-substituted 3-hydroxy-4-oxo-1,4-dihydroquinolines[J]. Tetrahedron Lett, 2016, 57(9): 1022-1026.
[24]SHMIDTM S, PERILLO I A, GONZÁLEZ M, et al. Reaction of isatin with alkylating agents with acidic methylenes[J]. Tetrahedron Lett, 2012, 53(20): 2514-2517.
[25]FENG L S, LIU M L, ZHANG S, et al. Synthesis and in vitro antimycobacterial activity of 8-OCH3 ciprofloxacin methylene and ethylene isatin derivatives[J]. Eur J Org Chem, 2011, 46(1): 341-348.